Filip Stefaniak

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Publications

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PubMed

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2021 AnnapuRNA: A scoring function for predicting RNA-small molecule binding poses

Topics:

graphical abstract

Filip Stefaniak, Janusz M Bujnicki
AnnapuRNA: A scoring function for predicting RNA-small molecule binding poses, February 1, 2021 | DOI: journal.pcbi.1008309

IF: 4.700

AnnapuRNA repository: github

2020 Luciferase reporter assay for small-molecule inhibitors of MIR92b-3p function: Screening cyanopeptolins produced by Nostoc from the Baltic Sea

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graphical abstract

Paweł Brzuzan, Hanna Mazur-Marzec, Maciej Florczyk, Filip Stefaniak, Anna Fidor, Robert Konkel, Maciej Woźny
Luciferase reporter assay for small-molecule inhibitors of MIR92b-3p function: Screening cyanopeptolins produced by Nostoc from the Baltic Sea
Toxicology in Vitro, 2020, Volume 68, 104951 | DOI: 10.1016/j.tiv.2020.104951

IF: 2.959; 5-Year IF:

2020 RNAProbe: a web server for normalization and analysis of RNA structure probing data

Topics:

graphical abstract

Tomasz K Wirecki, Katarzyna Merdas, Agata Bernat, Michał J Boniecki, Janusz M Bujnicki, and Filip Stefaniak
RNAProbe: a web server for normalization and analysis of RNA structure probing data
Nucleic Acids Research, 2020, Volume 48, Issue W1, Pages W292–W299 | DOI: 10.1093/nar/gkaa396

IF: 11.501; 5-Year IF: 11.797

The web server described in the paper: https://rnaprobe.genesilico.pl/

2020 Benzoxazepine-Derived Selective, Orally Bioavailable Inhibitor of Human Acidic Mammalian Chitinase

Topics:

Gleb Andryianau, Michal Kowalski, Michal C. Piotrowicz, Adam A. Rajkiewicz, Barbara Dymek, Piotr L. Sklepkiewicz, Elzbieta Pluta, Filip Stefaniak, Wojciech Czestkowski, Sylwia Olejniczak, Marzena Mazur, Piotr Niedziejko, Robert Koralewski, Krzysztof Matyszewski, Mariusz Gruza, Agnieszka Zagozdzon, Magdalena Salamon, Aleksandra Rymaszewska, Mikolaj Welzer, Karolina Dzwonek, Jakub Golab, Jacek Olczak, Agnieszka Bartoszewicz, and Adam Golebiowski

Benzoxazepine-Derived Selective, Orally Bioavailable Inhibitor of Human Acidic Mammalian Chitinase

ACS Med. Chem. Lett. 2020, 11, 6, Pages 1228–1235 | DOI: 10.1021/acsmedchemlett.0c00092

IF: 3.975 (2019)

2019 Development of Dual Chitinase Inhibitors as Potential New Treatment for Respiratory System Diseases

Topics:

Marzena Mazur, Barbara Dymek, Robert Koralewski, Piotr Sklepkiewicz, Sylwia Olejniczak, Marcin Mazurkiewicz, Michał Piotrowicz, Magdalena Salamon, Karol Jędrzejczak, Agnieszka Zagozdzon, Wojciech Czestkowski, Krzysztof Matyszewski, Bartłomiej Borek, Agnieszka Bartoszewicz, Elżbieta Pluta, Aleksandra Rymaszewska, Witold Mozga, Filip Stefaniak, Paweł Dobrzański, Karolina Dzwonek, Jakub Golab, Adam Golebiowski, and Jacek Olczak

Development of Dual Chitinase Inhibitors as Potential New Treatment for Respiratory System Diseases

Journal of Medicinal Chemistry, 62 (15), 2019, Pages 7126-7145 | DOI: 10.1021/acs.jmedchem.9b00681

IF: 6.205 (2019)

2019 Structural bases of peptidoglycan recognition by lysostaphin SH3b domain

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graphical abstract

Paweł Mitkowski, Elżbieta Jagielska, Elżbieta Nowak, Janusz M. Bujnicki, Filip Stefaniak, Dorota Niedziałek, Matthias Bochtler & Izabela Sabała

Structural bases of peptidoglycan recognition by lysostaphin SH3b domain

Scientific Reports, volume 9, Article number: 5965, 2019, Pages: tba | DOI: 10.1038/s41598-019-42435-z

IF: 4.122; 5-Year IF: 4.609

2018 Human RNA cap1 methyltransferase CMTr1 cooperates with RNA helicase DHX15 to modify RNAs with highly structured 5′ termini

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Diana Toczydlowska-Socha, Magdalena M. Zielinska, Malgorzata Kurkowska, Astha, Catarina F. Almeida, Filip Stefaniak, Elzbieta Purta, Janusz M. Bujnicki

Phil. Trans. R. Soc. B 2018 373, 20180161, 2018| DOI: 10.1098/rstb.2018.0161

IF: 5.666 (2017); 5-Year IF: 7.192

Visible also as: D Toczydlowska-Socha, M Kurkowska, M Zielinska, A Joshi, C Almeida, E Purta, F Stefaniak, J Bujnicki, FEBS OPEN BIO 9, 121-122, 2019.

2019 (conference paper) Riboswitch-ligand structure determination using an integrative structural biology approach

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A Ponce-Salvatierra, R Pluta, E Skowronek, M Orlowska, B Baginski, M Kurkowska, E Purta, P Ghosh, T Wirecki, F Stefaniak, JM Bujnicki

FEBS OPEN BIO, 9, 243-243, 2019.

2018 Synthesis and characterization of novel classes of PDE10A inhibitors - 1H-1,3-benzodiazoles and imidazo[1,2-a]pyrimidines

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graphical abstract

Rafał Moszczyński-Pętkowski, Jakub Majer, Małgorzata Borkowska, Łukasz Bojarski, Sylwia Janowska, Mikołaj Matłoka, Filip Stefaniak, Damian Smuga, Katarzyna Bazydło, Krzysztof Dubiel, Maciej Wieczorek

European Journal of Medicinal Chemistry 155, 15 July, 2018, Pages 96-116 | DOI: 10.1016/j.ejmech.2018.05.043

IF: 4.519; 5-Year IF: 4.187

2018 Discovery of selective, orally bioavailable inhibitor of mouse chitotriosidase.

Topics:

graphical abstract

Mazur M, Bartoszewicz A, Dymek B, Salamon M, Andryianau G, Kowalski M, Olejniczak S, Matyszewski K, Pluta E, Borek B, Stefaniak F, Zagozdzon A, Mazurkiewicz M, Koralewski R, Czestkowski W, Piotrowicz M, Niedziejko P, Gruza MM, Dzwonek K, Golebiowski A, Golab J, Olczak J

Bioorg Med Chem Lett. Volume 28, Issue 3, 1 February 2018, Pages 310-314 | DOI: 10.1016/j.bmcl.2017.12.047

IF: 2.454; 5-Year IF: 2.286

2018 Novel inhibitors of the rRNA ErmC′ methyltransferase to block resistance to Macrolides, Lincosamides, Streptogramine B antibiotics

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graphical abstract

Foik IP, Tuszynska I, Feder M, Purta E, Stefaniak F, Bujnicki JM
Eur J Med Chem Volume 146, 25 February 2018, Pages 60-67 | DOI: 10.1016/j.ejmech.2017.11.032

IF: 4.519; 5-Year IF: 4.187

2018 RNArchitecture: a database and a classification system of RNA families, with a focus on structural information

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graphical abstract

Boccaletto P, Magnus M, Almeida C, Zyla A, Astha, Pluta R, Baginski B, Jankowska E, Dunin-Horkawicz S, Wirecki T, Boniecki M, Stefaniak F, Bujnicki JM

Nucleic Acids Res. 2018 Jan 4;46(D1):D202-D205. | DOI: 10.1093/nar/gkx966

IF: 10.162

2018 Exploring Baltic Sea cyanobacteria for small-molecule inhibitors of microRNA function: a project description

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graphical abstract

Paweł Brzuzan, Hanna Mazur Marzec, Filip Stefaniak, Maciej Woźny, Maciej Florczyk

ENVIRONMENTAL BIOTECHNOLOGY 14 (1) 2018; Pages 1-4| DOI: 10.14799/ebms301 (doesn't work for some reasons...)

2016 Molecularly Imprinted Polymer (MIP) Film with Improved Surface Area Developed by Using Metal-Organic Framework (MOF) for Sensitive Lipocalin (NGAL) Determination

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Zofia Iskierko, Piyush Sindhu Sharma, Daniel Prochowicz, Krzysztof Fronc, Francis D'Souza, Diana Toczydlowska, Filip Stefaniak, Krzysztof Noworyta,

ACS Appl. Mater. Interfaces, 2016, 8 (31), pp 19860–19865 | DOI: 10.1021/acsami.6b05515

IF: 7.504

2015 Prediction of compounds activity in nuclear receptor signaling and stress pathway assays using machine learning algorithms and low dimensional molecular descriptors

Topics:

pipeline

Filip Stefaniak
Front. Environ. Sci., 01 December 2015 | DOI: 10.3389/fenvs.2015.00077

IF: 2.749

2015 Modeling of ribonucleic acid–ligand interactions

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Filip Stefaniak, Ewa Chudyk (Joint First Authorship), Michael Bodkin, Wayne Dawson, Janusz M. Bujnicki
WIREs Comput Mol Sci 2015, 5:425–439. | DOI: 10.1002/wcms.1226

IF: 14.016

2015 Discovery of TRAF-2 and NCK-interacting kinase (TNIK) inhibitors by ligand-based virtual screening methods

Topics:

TNIK cover

Anna Bujak, Filip Stefaniak (Joint First Authorship), Daria Zdzalik, Paulina Grygielewicz, Barbara Dymek, Marcin Zagozda, Pawel Gunerka, Monika Lamparska-Przybysz, Krzysztof Dubiel, Maciej Wieczoreka and Karolina Dzwonek
MedChemComm 6 (8), 2015, 1564-1572 | DOI: 10.1039/C5MD00090D

IF: 2.608